Design and Exploratory Neuropharmacological Evaluation of Novel Thyrotropin-Releasing Hormone Analogs and Their Brain-Targeting Bioprecursor Prodrugs (open access)

Design and Exploratory Neuropharmacological Evaluation of Novel Thyrotropin-Releasing Hormone Analogs and Their Brain-Targeting Bioprecursor Prodrugs

Paper describes novel and metabolically stable analogs derived from thyrotropin-releasing hormone (TRH) by replacing its amino-terminal pyroglutamyl (pGlu) residue with pyridinium-containing moieties.
Date: May 22, 2013
Creator: Prokai-Tatrai, Katalin; Nguyen, Vien; Szarka, Szabolcs; Konya, Krisztina & Prókai, László, 1958-
System: The UNT Digital Library